The Laboratory tubes

Samfura

Pimobendan 74150-27-9 Metabolism PDE inhibitor

Takaitaccen Bayani:

Sunan samfur:Pimobendan
Makamantuwa:4,5-Dihydro-6-[2- (4-methoxyphenyl) -1H-benzimizol-6-yl] -5-methyl-3 (2H) -pyridazinone
Lambar CAS:74150-27-9
inganci:USP43
Tsarin kwayoyin halitta:Saukewa: C19H18N4O2
Nauyin kwayoyin halitta:334.37


Cikakken Bayani

Tags samfurin

Biya:T/T, L/C
Asalin samfur:China
Tashar Jirgin Ruwa:Beijing/Shanghai/Hangzhou
Oda (MOQ):1 g
Lokacin Jagora:3 kwanakin aiki
Ƙarfin samarwa:1kg/wata
Yanayin ajiya:Ajiye a wuri mai sanyi, busasshiyar wuri, zazzabin ɗaki.
Kunshin kayan:kwalba, kwalba
Girman kunshin:1g / gwangwani, 5/kwali, 10g/kwali, 50g / kwalban, 500g / kwalban
Bayanin aminci:UN 2811 6.1/PG 3

Pimobendan

Gabatarwa

Pimobendan, maganin dabbobi ne.Yana da mai ilimin calcium kuma mai zaɓin mai hanawa na phosphodiesterase 3 (PDE3) tare da ingantaccen tasirin inotropic da vasodilator.

Ana amfani da Pimobendan wajen kula da gazawar zuciya a cikin karnuka, wanda aka fi sani da myxomatous mitral bawul cuta (wanda aka sani a baya da endocardiosis), ko dilated cardiomyopathy.Bincike ya nuna cewa a matsayin monotherapy, pimobendan yana ƙaruwa lokacin rayuwa kuma yana inganta rayuwa a cikin marasa lafiya na canine tare da raunin zuciya na biyu zuwa cututtukan mitral valve idan aka kwatanta da benazepril, mai hana ACE.

Musamman (USP43)

Abu

Ƙayyadaddun bayanai

Bayyanar

Farin fari ko dan kadan mai launin rawaya, hygroscopic

Mp

Kimanin 242 ℃

Solubility

A zahiri wanda ba a iya narkewa cikin ruwa, mai narkewa cikin yardar kaina a cikin dimethylformamide, mai narkewa a cikin acetone kuma cikin methanil.

Ganewa

Infrared absorption spectrophotometry, Kwatanta pimobendan CRS.

Lokacin riƙewa na babban kololuwar mafita na Samfurin ya yi daidai da na daidaitaccen bayani na hannun jari, kamar yadda aka samu a cikin gwajin ƙazantattun kwayoyin halitta.

Karfe masu nauyi

≤10pm

Granularity

P90 ≤ 25μm

Girman barbashi

20-80 guda

Ragowar kaushi

≤ 500ppm

Ruwa

≤ 1.0%

Assay

98.0% ~ 102.0%

Sulfate ash

0.10%

Abubuwan da ke da alaƙa (HPLC)

rashin tsarki A

0.10%

rashin tsarki B

0.10%

Duk wani kazanta

0.10%

Jimlar ƙazanta

0.20%


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